Cyproterone + Ethinyl Estradiol
Uses of Cyproterone + Ethinyl Estradiol
Cyproterone + Ethinyl Estradiol is used to treat moderate to severe acne and excessive hair growth (hirsutism) caused by high androgen levels in women.
This combination is commonly used for:
• Androgen-related acne: Reduces acne caused by excess androgen (male hormone) activity in women.
• Hirsutism: Reduces excessive hair growth on the face and body linked to high androgen levels.
• Polycystic ovary syndrome (PCOS): Manages symptoms associated with PCOS, such as acne and excess hair growth, when these are related to androgen excess.
• Contraception: Provides effective contraception when taken as prescribed.
Side effects of Cyproterone + Ethinyl Estradiol
Nausea
Headaches
Breast tenderness
Weight changes
Mood changes
How Cyproterone + Ethinyl Estradiol works
Cyproterone + Ethinyl Estradiol works through two hormonal actions that together reduce androgen-related symptoms and prevent pregnancy.
Cyproterone is an anti-androgen. It blocks androgen receptors in the skin and hair follicles, reducing the effects of male hormones that cause acne and excess hair growth.
Ethinyl Estradiol is a synthetic form of oestrogen. It increases the level of a protein that binds to androgens in the blood, which further reduces their activity, and it also prevents ovulation, providing contraceptive protection.
Together, these hormones reduce androgen-related skin and hair symptoms while offering reliable contraception.
Certified content
Written By
Doctor of Medicine
Reviewed By
BAMS, FMC, MD Resident
Expert Advice
Dosage Forms Available
- Cyproterone + Ethinyl Estradiol is available for use as oral tablets.
Age and Dose Restrictions
- This medicine is prescribed for women of reproductive age and is not recommended for use in children or men.
Contraindications
- Cyproterone + Ethinyl Estradiol is contraindicated in women who are pregnant or breastfeeding, smoke and are over 35 years old, have a history of blood clots, stroke, or heart attack, have severe liver disease, have certain types of migraine, have or have had breast cancer or other estrogen-sensitive cancers, and have undiagnosed vaginal bleeding.
Other Medications to Avoid
- Cyproterone + Ethinyl Estradiol may interact with certain antibiotics (such as rifampicin), antifungals (such as griseofulvin), anticonvulsants (like phenytoin, carbamazepine and phenobarbital), and HIV medications (such as ritonavir), and herbal supplements like St. John's Wort.
Overdose and Missed Dose
- Taking more than the prescribed dose may cause nausea, vomiting, breast tenderness, dizziness, fatigue, or withdrawal bleeding. If you notice these symptoms, consult your doctor immediately.
- If you miss a dose, take it as soon as you remember. If it is almost time for your next dose, skip the missed one. Do not take a double dose to make up for a missed one.
Management of Side Effects
Most side effects are temporary and generally harmless and resolve when discontinuing this medicine. However, if you experience any severe side effects or worsening of any of the symptoms, please consult your doctor.
- Drinking plenty of fluids can help manage side effects such as nausea.
- To manage headaches, try resting and taking a break from your regular activities.
- If you experience mood changes, try to rest and relax.
Use in Driving and Operating Machinery
- Cyproterone + Ethinyl Estradiol may cause dizziness or fatigue. If you experience these side effects, avoid driving or operating heavy machinery.
Use in Pregnancy and Lactation
- Cyproterone + Ethinyl Estradiol is not recommended during pregnancy or breastfeeding. If you are pregnant, planning to become pregnant, or breastfeeding, consult your doctor before using this medication.
Caution in Other Conditions
- Women with a history of liver disease or cancer should use Cyproterone + Ethinyl Estradiol with caution. Also, women with a history of blood clots or stroke should consult their doctor before using this medication.
Special Dietary and Lifestyle Recommendations
- Aim to maintain a healthy weight as being overweight can increase the risk of side effects.
- Include plenty of fruits and vegetables in your diet to keep your skin healthy.
- Limit alcohol consumption as it can increase the risk of side effects.
Frequently asked questions
Is Cyproterone + Ethinyl Estradiol a steroid?
Yes, Cyproterone + Ethinyl Estradiol is a combination of two hormones-cyproterone, an anti-androgen, and ethinyl estradiol, a form of oestrogen, both of which are types of steroids.
Does Cyproterone + Ethinyl Estradiol have any effect on sleep?
There is no direct evidence to suggest that Cyproterone + Ethinyl Estradiol impacts sleep. However, changes in hormone levels can sometimes indirectly influence sleep patterns. If you notice any significant changes in your sleep, consult your doctor.
Will Cyproterone + Ethinyl Estradiol affect fertility?
Cyproterone + Ethinyl Estradiol has contraceptive effects and prevents ovulation. Thus, it can affect fertility during its use. However, normal fertility is expected to return after discontinuation of the medication.
Are there any particular dietary restrictions while taking Cyproterone + Ethinyl Estradiol?
No specific dietary restrictions are mentioned in conjunction with the use of Cyproterone + Ethinyl Estradiol. However, maintaining a balanced diet is always beneficial for overall health.
Is it safe to take Cyproterone + Ethinyl Estradiol daily?
Yes, it is safe to take Cyproterone + Ethinyl Estradiol daily as prescribed by your doctor for the treatment of conditions like acne or hirsutism or as a contraceptive.
How much time does Cyproterone + Ethinyl Estradiol take to show its effects?
Improvements in conditions like acne are usually seen after about 3 months of consistent use. Maximum benefits are seen after about 6 months.
Is Cyproterone + Ethinyl Estradiol available over the counter, or do I need a prescription?
Cyproterone + Ethinyl Estradiol is a prescription medication and is not available over the counter.
What is the use of Cyproterone + Ethinyl Estradiol?
Cyproterone + Ethinyl Estradiol is used to manage hormone-related conditions in women, such as acne, excessive hair growth (hirsutism), and symptoms of polycystic ovary syndrome (PCOS). It works by reducing the effect of male hormones (androgens) in the body and also helps regulate the menstrual cycle. In some cases, it may also be prescribed for contraception when these hormonal conditions are present.
Cyproterone + Ethinyl Estradiol in other salts
List of medicines for Cyproterone + Ethinyl Estradiol
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